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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T68599 | Orphenadrine | Orphenadrine (free base) | Sodium Channel , NMDAR , AChR |
Orphenadrine is a noncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist that inhibits clonal HERG channels in a concentration-dependent manner, producing an IC of 0.85 μM in HEK cells.Orphenadrine is an antagoni... | |||
T70487 | Tofenacin (free base) | ||
Tofenacin (free base) is an antidepressant drug with a tricyclic-like structure. It acts as a serotonin-norepinephrine reuptake inhibitor, and based on its close relation to orphenadrine, may also possess anticholinergic... |